Our potent and selective hA3 adenosine receptor fluorescent antagonist shows a high affinity and selectivity for hA3 receptor over the other receptor subtypes (Ki = 6.13 nM for A3 receptor in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

CELT-071 hA3 adenosine receptor fluorescent antagonist (589/616)

10 μg vial that allows to prepare 86 mL of 100 nM working solution to test A3R.

Working concentration might differ among assay designs

432,00

Available on back-order