Our potent and selective hα1A  adrenergic receptor fluorescent antagonist shows high affinity for α1A adrenergic receptor (Ki = 28.3 nM measured in radioligand binding assay) and selectivity over α2A (Ki = 1081 nM measured in radioligand binding assay). It is potentially suitable for fluorescence-based assays such as confocal microscopy or high content screening.

CELT-030 hα1A adrenergic receptor fluorescent antagonist (646/662)

10 µg vial that allows to prepare 83 mL of 100 nM working solution to test α1AR.

Working concentration might differ among assay designs
Our CELT-030 product has been developed to meet the needs of researchers in a variety of fields, enabling the study of α1A adrenergic receptors with greater accuracy and precision.

432,00