Potent and selective hA₁ adenosine receptors fluorescent antagonist (560/571)

Our potent and selective hA₁ adenosin receptor fluorescent antagonist shows affinity and selectivity for hA₁ (K_i = 26.2 nM in radioligand binding assays). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.