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Our potent and partially selective hA1 adenosine receptor fluorescent antagonist shows higher affinity for hA1 (Ki = 8.60 nM) compared to hA2A, hA2B and hA3 adenosine receptors (Ki = 98.38 nM, 72.24 nM and 231.01 nM respectively in radioligand binding assays). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

CELT-360 hA1 adenosine receptor fluorescent antagonist (646/662)

10 µg vial that allows to prepare 79 mL of 100 nM working solution to test A1R.

Working concentration might differ among assay designs

432,00