Our potent hA_2B/A₃ adenosine receptor fluorescent antagonist shows high affinity for hA_2B and A₃ receptor (K_i = 35.6 nM and 45.7 nM respectively in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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