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Our potent and selective hα1A adrenergic receptor fluorescent antagonist shows high affinity for α1A adrenergic receptor (Ki = 5 nM measured in radioligand binding assay) and selectivity over α2A (15% of displacement at 1 μM in radioligand binding assay). It is potentially suitable for fluorescence-based assays such as confocal microscopy, high content screening or fluorescence polarization.

CELT-033 hα1A adrenergic receptor fluorescent antagonist (560/571)

This product is available in a 10 µg vial that allows you to prepare 76 mL of 100 nM working solution to test α1AR.

The working concentration might differ among assay designs
Our CELT-033 ligand has been specifically designed for high potency and selectivity. It has a high affinity for α1A receptor and may be suitable for fluorescence-based assays.

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